bcx 1812 has been researched along with (3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone in 1 studies
Studies (bcx 1812) | Trials (bcx 1812) | Recent Studies (post-2010) (bcx 1812) | Studies ((3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone) | Trials ((3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone) | Recent Studies (post-2010) ((3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone) |
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25 | 1 | 12 | 38 | 1 | 15 |
Protein | Taxonomy | bcx 1812 (IC50) | (3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone (IC50) |
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Histone deacetylase 3 | Homo sapiens (human) | 0.0151 | |
Cytochrome P450 1A2 | Homo sapiens (human) | 0.011 | |
Cytochrome P450 3A4 | Homo sapiens (human) | 0.011 | |
Cytochrome P450 2D6 | Homo sapiens (human) | 0.034 | |
Cytochrome P450 2C9 | Homo sapiens (human) | 0.034 | |
Tissue factor | Homo sapiens (human) | 0.175 | |
Cytochrome P450 2B6 | Homo sapiens (human) | 0.034 | |
Cytochrome P450 3A5 | Homo sapiens (human) | 0.011 | |
Cytochrome P450 2C19 | Homo sapiens (human) | 0.011 | |
Histone deacetylase 4 | Homo sapiens (human) | 1.0335 | |
Histone deacetylase 1 | Homo sapiens (human) | 0.0227 | |
Histone deacetylase 7 | Homo sapiens (human) | 0.014 | |
Histone deacetylase 2 | Homo sapiens (human) | 0.0185 | |
Polyamine deacetylase HDAC10 | Homo sapiens (human) | 0.014 | |
Histone deacetylase 11 | Homo sapiens (human) | 0.014 | |
Histone deacetylase 8 | Homo sapiens (human) | 0.2852 | |
Histone deacetylase | Cryptosporidium parvum | 0.001 | |
Histone deacetylase | Cryptosporidium parvum | 0.001 | |
Histone deacetylase 6 | Homo sapiens (human) | 1.4663 | |
Histone deacetylase 9 | Homo sapiens (human) | 0.014 | |
Histone deacetylase 5 | Homo sapiens (human) | 0.014 | |
Histone deacetylase | Plasmodium falciparum (malaria parasite P. falciparum) | 0.001 | |
Nuclear receptor corepressor 2 | Homo sapiens (human) | 0.0193 |
Timeframe | Studies, this research(%) | All Research% |
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pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 1 (100.00) | 2.80 |
Authors | Studies |
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Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M | 1 |
1 other study(ies) available for bcx 1812 and (3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone
Article | Year |
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In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries | 2023 |